Enalapril Maleate
abẹlẹ
Enalapril Maleate
Apejuwe
Enalapril (maleate) (MK-421 (maleate)), metabolite ti nṣiṣe lọwọ ti enalapril, jẹ inhibitor enzymu iyipada angiotensin (ACE).
Ninu Vivo
Enalapril (MK-421) jẹ oogun oogun ti o jẹ ti ẹgbẹ inhibitor enzymu iyipada angiotensin (ACE) ti awọn oogun. O ti ni metabolized ni iyara ninu ẹdọ si enalaprilat lẹhin iṣakoso ẹnu. Enalapril (MK-421) jẹ apaniyan ti o lagbara, ifigagbaga ti ACE, enzymu ti o ni iduro fun iyipada angiotensin I (ATI) si angiotensin II (ATII). ATII ṣe ilana titẹ ẹjẹ ati pe o jẹ paati bọtini ti eto renin-angiotensin-aldosterone (RAAS). Enalapril le ṣee lo lati ṣe itọju pataki tabi haipatensonu iṣan iṣan ati ikuna ọkan iṣọn-alọ ọkan.
Ibi ipamọ
Lulú | -20°C | 3 odun |
4°C | ọdun meji 2 | |
Ni epo | -80°C | osu 6 |
-20°C | osu 1 |
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